Pain Killer Flupirtine Maleate Powder Flupirtine Maleate

• Customization: Available
• CAS No.: 75507-68-5
• Formula: C19h21fn4o6
• Model NO.: QS-Flupirtine Maleate
• EINECS: 278-225-0
• Packaging Material: Negotiable
• Storage Method: Normal
• Shelf Life: >12 Months
• Nutrient Composition: Flupirtine Maleate
• Resource: Flupirtine Maleate
• The content of active substances: >99%
• Product Name: Flupirtine Maleate
• Name: Flupirtine Maleate Powder
• Appearance: White Powder
• Colour: White
• Grade: Pharmaceutical Grade
• Assay: >99%
• Application: API
• Specific: COA
• Test Method: HPLC
• MW: 420.39
• Mf: C19h21fn4o6
• Boiling Point: 434.9
• Melting Point: 186-188c
• Certification: GMP, Hse, ISO 9001, USP, Bp
• Suitable for: Elderly, Children, Adult
• Transport Package: Negotiable
• Specification: >99%
• Trademark: QS-Flupirtine Maleate
• Origin: Xian
• Production Capacity: 1000kg/Month

Product Description

Hot Sale Relieve Pain Flupirtine Maleate 99% Flupirtine Maleate

Product Description

Product Details

Product Name	Flupirtine Maleate
Appearance	Flupirtine Maleate Powder
Assay	>99%
MW	420.39
MF	C19h21fn4o6
Boiling Point	434.9
Melting Point	186-188c

Flupiritine malate is a non opioid central analgesic that is a selective neuronal potassium channel opener and possesses NMDA receptor antagonist properties. It is mainly administered orally and has significant analgesic effects, especially in relieving pain caused by various reasons.
Fluoxetine maleate (CAS number: 75507-68-5) is the maleic acid salt form of fluoxetine and belongs to the central non opioid analgesic class. It has analgesic and muscle relaxant effects by activating neuronal potassium channels (Kv7), regulating NMDA receptor activity, and inhibiting glutamate release. It is mainly used to treat acute pain such as postoperative pain and chronic pain such as neuropathic pain, osteoarthritis, and can relieve pain related muscle tension. In terms of pharmacokinetics, the oral bioavailability of the drug is 50% -70%, and the maleic acid salt structure may enhance solubility and absorption efficiency; Metabolized by the liver as inactive products and excreted by the kidneys.

Application&Function

Pharmacological effects and uses
Flupiritine malate exerts analgesic effects by opening neuronal potassium channels and inhibiting NMDA receptors. Its analgesic effect is similar to , but the intensity is weaker, about 50% of . In addition, it also has muscle relaxation and neuroprotective effects.

Specification